CAS number：861393-28-4 molecular formula：C26H30N6O3
A-740003是P2X7受体选择性抑制剂，对鼠和人P2X7受体的IC50分别为18和40 nM。 A-740003 是一种高度仿射和选择性 P2X7 受体拮抗剂，最适合于放射性示踪剂进展，用于正电子发射断层扫描神经炎症成像。 A-740003 是一种有效的，选择性的，竞争性的 P2X7 receptor 拮抗剂，抑制大鼠和人的 P2X7 受体，IC50 值分别为 18 和 40 nM。 A-740003 is potent, selective and competitive P2X7 receptor antagonist (IC50 values are 18 and 40 nM for rat and human receptors respectively). A potent, selective and competitive P2X7 receptor antagonist
| Chinese alias | N-(1-{[(氰亚胺基)(5-喹啉氨基)甲基] 氨基 }-2,2-二甲基丙基)-2-(3,4-二甲氧基苯基)乙酰胺 | ||
| English alias | N-[1-[(E)-[(cyanoamino)-(quinolin-5-ylamino)methylidene]amino]-2,2-dimethylpropyl]-2-(3,4-dimethoxyphenyl)acetamide | ||
| CAS number | 861393-28-4 | molecular formula | C26H30N6O3 |
| molecular weight | 474.55 g/mol | Exact mass | - |
| PSA | 121.000 Ų | logp | 4.600 |
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