•蛋白-蛋白相互作用(PPI)代表了细胞内外的一大类治疗靶标。许多蛋白质-蛋白质相互作用(PPI)的抑制剂已成为潜在的抗癌药物; •173种蛋白与蛋白相互作用(PPI)抑制剂的独特集合,适用于高通量筛选(HTS)和高内涵筛选(HCS); •靶点包括PD-1/PD-L1, BCL family, Bromodomains, MDM2, HIV integras等; •某些化合物已被FDA批准; •结构多样,具有药用活性且可渗透细胞; •提供丰富的文档信息,包括化合物结构和生物活性信息; •验证NMR和HPLC以确保高纯度。 详细信息 配制:
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Protein-protein Interaction Inhibitor Library
CAS number:unknown molecular formula:
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| Chinese alias | - | ||
| English alias | - | ||
| CAS number | unknown | molecular formula | |
| molecular weight | - | Exact mass | - |
| PSA | - | logp | - |
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