CAS number：1637770-13-8 molecular formula：C25H22N4O
GS-626510 is a potent, and orally active BET family bromodomains inhibitor, with K d values of 0.59-3.2 nM for BRD2/3/4, with IC 50 values of 83 nM and 78 nM foe BD1 and BD2 , respectively Form:Solid IC50& Target:BRD2 0.59-2.5 nM (Kd) BRD3 0.65-0.66 nM (Kd) BRD4 1.3-3.2 nM (Kd) BD1 83 nM (IC 50 ) BD2 78 nM (IC 50 )
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| CAS number | 1637770-13-8 | molecular formula | C25H22N4O |
| molecular weight | 394.47 g/mol | Exact mass | ≥99% |
| PSA | - | logp | - |
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