CAS number：315694-89-4 molecular formula：C17H12N2O2
TC-DAPK 6 is a potent, ATP-competitive, and highly selective DAPK inhibitor ( IC 50 =69 and 225 nM against DAPK1 and DAPK3 , respectively, with 10 μM ATP). In Vitro TC-DAPK 6 is found to be the most potent Death-associated protein kinase (DAPK) inhibitor with enzyme selectivity. When assayed with 10 μM ATP, the IC 50 values for DAPK1 and DAPK3 are 69 and 225 nM, respectively. TC-DAPK 6 also inhibits p70S6K (1 μM Form:Solid IC50& Target:IC50: 69 nM (DAPK1), 225 nM (DAPK3)
| Chinese alias | - | ||
| English alias | EX-A2167 | Z56820688 | EN300-260619 | AC-35960 | EN300-7536106 | 2-(2-phenylethenyl)-4-[(pyridin-3-yl)methylidene]-4,5-dihydro-1,3-oxazol-5-one | TC-DAPK-6 | (E)-4-(pyridin-3-ylmethylene)-2-((E)-styryl)oxazol-5(4H)-one | HY-15513 | 4-(pyridin-3-ylmethylen | ||
| CAS number | 315694-89-4 | molecular formula | C17H12N2O2 |
| molecular weight | 276.29 g/mol | Exact mass | ≥98% |
| PSA | 51.600 Ų | logp | 2.9 |
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