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BPR1K871

CAS number:2443767-35-7    molecular formula:C25H28ClN7O2S

overview

compound introduction

Information BPR1K871 (DBPR114) is a potent and selective dual inhibitor of FLT3 and AURKA with IC50 of 19 nM and 22 nM, respectively. BPR1K871 (DBPR114) acts as a preclinical development candidate for anti-cancer therapy.

Specs

Chinese alias-
English aliasDBPR114
CAS number2443767-35-7molecular formulaC25H28ClN7O2S
molecular weight526.1 g/molExact mass-
PSA133.000 Ųlogp4.8

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