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PTC-209 HBr

CAS number:1217022-63-3    molecular formula:C17H14Br3N5OS

overview

compound introduction

PTC-209 HBr 是PTC-209的氢溴酸盐 , 这是一种强效的选择性的BMI-1抑制剂,其IC50为0.5 μM, 可以不可逆的减少癌起始细胞(CICs)。

Specs

Chinese alias-
English aliasPTC-209 hydrobromide | N-(2,6-dibromo-4-methoxyphenyl)-4-(2-methylimidazo[1,2-a]pyrimidin-3-yl)thiazol-2-amine hydrobromide
CAS number1217022-63-3molecular formulaC17H14Br3N5OS
molecular weight576.1 g/molExact mass≥98%
PSA92.600 Ųlogp-

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