CAS number：1609564-75-1 molecular formula：C30H32N4O5S
DY268 是法尼样X受体 (FXR) 的拮抗剂(在 time-resolved FRET 分析中，IC50=7.5 nM)。在细胞分析中，它抑制 FXR 反式激活。IC50 值为 468 nM。 Product description DY268 is a farnesoid X receptor (FXR) antagonist (IC50=7.5 nM in a time-resolved FRET assay). It inhibits FXR transactivation in a cell-based assay with an IC50 value of 468 nM.
| Chinese alias | 1-[(3-甲氧基苯基)甲基] -N-[4-甲基-3-(4-吗啉基磺酰基)苯基] -3-(4-甲基苯基)-1H-吡唑-4-羧酰胺 | ||
| English alias | 1-[(3-Methoxyphenyl)methyl]-N-[4-methyl-3-(4-morpholinylsulfonyl)phenyl]-3-(4-methylphenyl)-1H-pyrazole-4-carboxamide | ||
| CAS number | 1609564-75-1 | molecular formula | C30H32N4O5S |
| molecular weight | 560.66 g/mol | Exact mass | ≥98%(HPLC) |
| PSA | 111.000 Ų | logp | 3.8 |
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