Etoperidone 是一种抗抑郁剂,是一种具有口服活性的血清素 (serotonin) 和去甲肾上腺素 (nor-adrenaline) 再摄取拮抗剂。Etoperidone 对5-HT2受体、α1-肾上腺素受体 (α1-adrenergic receptor)、5-HT1A受体和 α2-肾上腺素受体 (α2-adrenergic receptor) 的Kd值分别为 36 nM、38 nM、85 nM 和 570 nM。
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Etoperidone
CAS number:52942-31-1 molecular formula:C19H28ClN5O
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| Chinese alias | - | ||
| English alias | - | ||
| CAS number | 52942-31-1 | molecular formula | C19H28ClN5O |
| molecular weight | 377.9 g/mol | Exact mass | - |
| PSA | 42.400 Ų | logp | 3 |
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