T3Inh-1 是一种有效且选择性的ppGalNAc-T3抑制剂(IC50=7 μM)。T3Inh-1 可降低组织细胞和小鼠体内的 FGF23 激素水平,且不会产生任何毒副作用。T3Inh-1 还可以预防乳腺癌细胞。ppGalNAc-T3 酶至少涉及两种重要的医学途径:癌症转移和FGF23的稳定 (调节血液中的磷酸盐水平)。
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4-[(6-nitroquinolin-4-yl)amino]-N-[4-(pyridin-4-ylamino)phenyl]benzamide
CAS number:50440-30-7 molecular formula:
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| Chinese alias | - | ||
| English alias | - | ||
| CAS number | 50440-30-7 | molecular formula | |
| molecular weight | 476.500 g/mol | Exact mass | ≥98% |
| PSA | 125.000 Ų | logp | 4.9 |
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