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DRAK2-IN-1

CAS number:871837-60-4    molecular formula:C21H20N4O3

overview

compound introduction

DRAK2-IN-1, compound 16, is a potent, selective and ATP-competitive DRAK2 inhibitor with IC 50 and K i values of 3 nM and 0.26 nM, respectively.DRAK2-IN-1 also has inbitory effect on DRAK1 ( IC 50 =51 nM) Form:Solid IC50& Target:IC50: 3 nM (DRAK2),51 nM (DRAK1),1.8 μM (DRPK2),2.3 μM (DRAK2),1.8 μM (DRPK3)

Specs

Chinese alias-
English alias-
CAS number871837-60-4molecular formulaC21H20N4O3
molecular weight376.41 g/molExact mass≥99%
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