Pepstatin (Pepstatin A) Trifluoroacetate is a specific, orally active aspartic protease inhibitor produced by actinomycetes, with IC 50 s of 4.5 nM, 6.2 nM, 150 nM, 290 nM, 520 nM and 260 nM for hemoglobin-pepsin, hemoglobin-proctase, casein-pepsin, casei Appearance:Solid IC50& Target:IC50: 4.5 nM (Hemoglobin-pepsin), 6.2 nM (Hemoglobin-proctase), 150 nM (Casein-pepsin), 260 nM (Hemoglobin-acid protease), 290 nM (Casein-proctase), 520 nM (Casein-acid protease) In Vitro:Pepstatin (Pepstatin A) (7 μM; 48 h) affects the intracellular processing of HIV-specific gag protein. MCE has not independently confirmed the accuracy of these methods. They are for reference only. In Vivo:Pepstatin (Pepstatin A) has a very low toxicity, with LD 50 s of 1090mg/kg, 875mg/kg, 820mg/kg and 450mg/kg for mice, rats, rabbits, and dogs by i.p. route, and > 2000mg/kg for all species by oral route. Pepstatin (0.5-50mg/kg, p.o.) suppresses Biological Activity:Pepstatin (Pepstatin A) Trifluoroacetate is a specific, orally active aspartic protease inhibitor produced by actinomycetes, with IC 50 s of 4.5 nM, 6.2 nM, 150 nM, 290 nM, 520 nM and 260 nM for hemoglobin-pepsin, hemoglobin-proctase, casein-pepsin, casei
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Pepstatin Trifluoroacetate
CAS number：unknown molecular formula：C36H64F3N5O11
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| Chinese alias | 胃酶抑素三氟乙酸酯 | ||
| English alias | - | ||
| CAS number | unknown | molecular formula | C36H64F3N5O11 |
| molecular weight | 799.92 g/mol | Exact mass | ≥99% |
| PSA | - | logp | - |
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