Integrin Antagonists 27 is a small molecule integrin αvβ3 antagonist with binding affinity of 18 nM, as s novel anticancer agent.Target: Integrin in vitro: Integrin Antagonists 27 is treated with a panel of cancer cell-lines (breast cancer cell line MDA-MB-435, breast cancer cell lines MCF-7, mouse fibroblast NIH3T3, ovarian cancer cell line HEY, lung cancer cell line NCI-H1975) with all IC50 of >20 uM. Form:Solid
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Integrin Antagonists 27
CAS number:593274-97-6 molecular formula:C24H20N4O5
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| Chinese alias | 整合素拮抗剂 27 | ||
| English alias | - | ||
| CAS number | 593274-97-6 | molecular formula | C24H20N4O5 |
| molecular weight | 444.44 g/mol | Exact mass | ≥98% |
| PSA | - | logp | - |
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