Enpp-1-IN-2 (Compound C) is a potent ENPP1 (ectonucleotide pyrophosphatase/phosphodiesterase 1) inhibitor with IC 50 values of 0.26, 0.48 and 2.0 μM evaluated by means of TG-mAMP, pNP-TMP, and ATP assays, respectively. TG (Tokyo Green)-mAMP: a newly synthesized sensitive ENPP1 fluorescence probe Form:Solid IC50& Target:IC 50 : 0.26 μM (TG-mAMP assay), 0.48 μM (pNP-TMP assay), 2.0 μM (ATP assay)
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Enpp-1-IN-2
CAS number:2378640-92-5 molecular formula:C15H18N6
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| Chinese alias | - | ||
| English alias | Enpp-1-IN-2 | 6-[(3-aminophenyl)methyl]-N,N,5-trimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine | ENPP1 Inhibitor C | SCHEMBL24129143 | AKOS040755821 | MS-24013 | HY-139362 | Z4180066045 | ||
| CAS number | 2378640-92-5 | molecular formula | C15H18N6 |
| molecular weight | 282.34 g/mol | Exact mass | ≥99% |
| PSA | - | logp | - |
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