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BRD7-IN-1

CAS number:2448414-48-8    molecular formula:C22H28Cl2N4O3

overview

compound introduction

BRD7-IN-1, a modified derivative of BI7273 (BRD7/9 inhibitor), binds to a VHL ligand via a linker to form a PROTAC VZ185 (VZ185 against BRD7/9 with DC 50 s of 4.5 and 1.8 nM, respectively) Form:Solid IC50& Target:BRD7, BRD9

Specs

Chinese alias-
English alias-
CAS number2448414-48-8molecular formulaC22H28Cl2N4O3
molecular weight467.39 g/molExact mass≥99%
PSA-logp-

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