FLTX1 是一种荧光他莫昔芬 (Tamoxifen) 衍生物,可以在透化和非透化条件下特异性标记细胞内 Tamoxifen 结合位点 (雌激素受体)。FLTX1 在乳腺癌细胞中表现出 Tamoxifen 有效的抗雌激素特性。FLTX1 缺乏对子宫的雌激素激动作用。 Information FLTX1, a fluorescent Tamoxifen derivative, can specifically label intracellular Tamoxifen-binding sites (estrogen receptors) under permeabilized and non-permeabilized conditions. FLTX1 exhibits potent antiestrogenic properties of Tamoxifen in breast cancer cells.
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FLTX1
CAS number:1481401-71-1 molecular formula:C31H28N4O4
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| Chinese alias | - | ||
| English alias | - | ||
| CAS number | 1481401-71-1 | molecular formula | C31H28N4O4 |
| molecular weight | 520.6 g/mol | Exact mass | ≥98% |
| PSA | - | logp | - |
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