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LOXO-195 R racemate

CAS number:1350884-56-8    molecular formula:C20H21FN6O

overview

compound introduction

(3aR)-Selitrectinib ((3aR)-LOXO-195) 是Selitrectinib 的一种异构体。Selitrectinib (LOXO-195) 是一种二代原肌凝蛋白相关激酶(TRK)抑制剂,其对TRKA和TRKC的IC50值分别为 0.6 nM 和

Specs

Chinese alias-
English alias-
CAS number1350884-56-8molecular formulaC20H21FN6O
molecular weight380.4 g/molExact mass-
PSA75.400 Ųlogp2.000

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