5-HT2A/5-HT2C inverse agonist 1 is a potent and dual 5-HT2A and 5-HT2C receptor inverse agonist with a hERG inhibitions, thus avoiding cardiovascular risks. 5-HT2A/5-HT2C inverse agonist 1 shows significant antipsychotic efficacy in the MK-801 -induced mouse model. 5-HT2A/5-HT2C inverse agonist 1 is promising for research of psychosis.
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5-HT2A/5-HT2C inverse agonist 1
CAS number:2718990-76-0 molecular formula:C24H35N5O2
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| Chinese alias | - | ||
| English alias | - | ||
| CAS number | 2718990-76-0 | molecular formula | C24H35N5O2 |
| molecular weight | 425.57 g/mol | Exact mass | - |
| PSA | - | logp | - |
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