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Pdk4-IN-1

CAS number:2310262-10-1    molecular formula:C22H19N3O2

overview

compound introduction

PDK4-IN-1 是一种蒽醌衍生物,也是一种有效的,口服活性的丙酮酸脱氢酶激酶 4 (PDK4) 抑制剂,IC50值为 84 nM。PDK4-IN-1 有效抑制细胞转化和细胞增殖并诱导细胞凋亡 (apoptosis)。PDK4-IN-1 具有抗糖尿病,抗癌和抗过敏作用。

Specs

Chinese alias-
English alias-
CAS number2310262-10-1molecular formulaC22H19N3O2
molecular weight357.4 g/molExact mass≥98%
PSA64.000 Ųlogp2.800

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