CAS number：708991-09-7 molecular formula：C13H16N4O2S
YUKA1 is a potent and cell permeable Lysine demethylase 5A ( KDM5A ) inhibitor, with an IC 50 of 2.66 μM, less active on KDM5C (IC 50 , 7.12 μM), and is inactive on KDM5B, KDM6A or KDM6B. YUKA1 increases H3K4me3 levels in human cells with anti-cancer activity Form:Solid IC50& Target:KDM5
| Chinese alias | - | ||
| English alias | DTXSID101326169 | SCHEMBL17133087 | AKOS000623644 | SMR000288072 | 4-{[(3-methoxy-2-prop-2-enyloxyphenyl)methyl]amino}-1,2,4-triazole-3-thiol | YUKA1 | MLS000709605 | 4-[(3-methoxy-2-prop-2-enoxyphenyl)methylamino]-1H-1,2,4-triazole-5-thione | 4-({[3-meth | ||
| CAS number | 708991-09-7 | molecular formula | C13H16N4O2S |
| molecular weight | 292.36 g/mol | Exact mass | ≥99% |
| PSA | 90.200 Ų | logp | 1.800 |
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