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Morphiceptin

CAS number:74135-04-9    molecular formula:C28H35N5O5

overview

compound introduction

Morphiceptin is a potent and specific agonist for morphine (μ) receptors . Morphiceptin, as a synthetic peptide, is the amide of a fragment of the milk protein β-casein. Morphiceptin has morphinelike activities and is highly specific for morphine (μ) receptors but not for enkephalin (⸹) receptors In Vivo Morphiceptin potently inhibits the binding of [ 3 H]dihydromorphine, 125 I-labeled FK33824, and [ 3 H]naloxone to rat brain membrane preparations with a 50 percent inhibition concentration (IC 50 ) of about 20 nM . MCE has not independently confirmed the accuracy of these methods. They are for reference only. Form:Solid IC50& Target:μ Opioid Receptor/MOR

Specs

Chinese alias吗啡肽
English aliasb-Casomorphin-4-amide | MS-29674 | Morphiceptin | N-(1-{2-[Hydroxy(imino)methyl]pyrrolidin-1-yl}-1-oxo-3-phenylpropan-2-yl)-1-tyrosylpyrrolidine-2-carboximidic acid | beta-Casomorphin-4-amide | beta-Casomorphine(1-4) amide | CHEBI:177741 | L-Tyrosyl-L-pro
CAS number74135-04-9molecular formulaC28H35N5O5
molecular weight521.61 g/molExact mass≥99%
PSA159.000 Ųlogp1.300

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