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RG 13022

CAS number:149286-90-8    molecular formula:

overview

compound introduction

(Z)-RG-13022 是一种酪氨酸激酶 (TK) 抑制剂,优先抑制EGFRTK 活性,抑制EGF刺激的培养细胞生长。(Z)-RG-13022 对 HN5 细胞的 DNA 合成表现出 11 μM 的IC50,比 (E)-RG-13022 (IC50=38 μM) 强 3 倍以上。(Z)-RG-13022 可用于乳腺癌细胞的研究。

Specs

Chinese alias-
English alias-
CAS number149286-90-8molecular formula
molecular weight266.290 g/molExact mass-
PSA55.100 Ųlogp2.600

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