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Setrobuvir

CAS number:1071517-39-9    molecular formula:

overview

compound introduction

Setrobuvir (ANA598) 是一种口服活性的非核苷HCVNS5B聚合酶抑制剂。Setrobuvir 抑制 RNA 的从头合成 (RNA synthesis) 和引物延伸,IC50在 4~5 nM 之间。Setrobuvir 还显示出与 SARS-CoV-2RdRp的优异结合亲和力,并诱导 RdRp 抑制。

Specs

Chinese alias-
English alias-
CAS number1071517-39-9molecular formula
molecular weight560.600 g/molExact mass-
PSA162.000 Ųlogp1.700

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