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NAMPT inhibitor-linker 2

CAS number:2241014-82-2    molecular formula:C34H33FN6O5

overview

compound introduction

粉末-20°C 3年,4°C 2年在溶剂中-80°C 6个月,-20°C 1个月 Powder -20°C 3 years,4°C 2 years;In solvent -80°C 6 months,-20°C 1 month In vivo activity ADC-4 (20 mg/kg, i.v. for 28 days) is tolerated, and causes tumor stasis in mice bearing GIST-T1 cells In vitro activity ADC-4 exihibits potent activity against c-Kit expressing cell lines such as GIST-T1 and NCI-H526, with IC50s of

Specs

Chinese alias-
English alias-
CAS number2241014-82-2molecular formulaC34H33FN6O5
molecular weight624.66 g/molExact mass≥99%
PSA-logp-

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