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TrkA-IN-1

CAS number:1680179-43-4    molecular formula:C25H20N4O

overview

compound introduction

TrkA-IN-1 is a potent and selective Tropomyosin-related kinase A (TrkA) inhibitor with an IC 50 of 99 nM in a cell-based assay. TrkA-IN-1 has analgesic activity Form:Solid IC50& Target:TrkA 99 nM (IC 50 ) TrkB 81 μM (IC 50 ) TrkC 25 μM (IC 50 )

Specs

Chinese alias-
English alias-
CAS number1680179-43-4molecular formulaC25H20N4O
molecular weight392.45 g/molExact mass≥98%
PSA66.900 Ųlogp4.200

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