CAS number：1458630-17-5 molecular formula：C16H16N6•CF3CO2H
CHR-6494 TFA 是一种有效的选择性 haspin 抑制剂，IC50 值为 2 nM。CHR-6494 TFA 能够抑制组蛋白 H3T3 的磷酸化。CHR-6494 TFA 诱导黑色素瘤、乳腺癌等肿瘤细胞凋亡 (apoptosis)。CHR-6494 TFA 可用于癌症的研究。 Product description： CHR-6494 TFA is a potent inhibitor of haspin, with an IC50 of 2 nM. CHR-6494 TFA inhibits histone H3T3 phosphorylation. CHR-6494 TFA induces the apoptosis of cancer cells, including melanoma and breast cancer. CHR-6494 TFA can be used in the research of cancer.
| Chinese alias | 3-(1H-吲唑-5-基)-N-丙基咪唑并[1,2-b]哒嗪-6-胺三氟乙酸盐 | ||
| English alias | 3-(1H-Indazol-5-yl)-N-propylimidazo[1,2-b]pyridazin-6-amine trifluoroacetate | ||
| CAS number | 1458630-17-5 | molecular formula | C16H16N6•CF3CO2H |
| molecular weight | 406.36 g/mol | Exact mass | ≥98%(HPLC) |
| PSA | 108.000 Ų | logp | - |
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