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N-benzyl-2-chloro-N-[1-(4-morpholin-4-ylbenzoyl)azepan-4-yl]acetamide

CAS number:2143467-62-1    molecular formula:

overview

compound introduction

BPK-29 是一种特殊的配体,通过共价修饰 C274 来破坏非典型孤核受体NR0B1与RBM45,SNW1蛋白质的相互作用。BPK-29 损害KEAP1突变癌细胞的锚定独立生长。

Specs

Chinese alias-
English alias-
CAS number2143467-62-1molecular formula
molecular weight470.000 g/molExact mass≥99%
PSA53.100 Ųlogp3.700

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