BPK-29 是一种特殊的配体,通过共价修饰 C274 来破坏非典型孤核受体NR0B1与RBM45,SNW1蛋白质的相互作用。BPK-29 损害KEAP1突变癌细胞的锚定独立生长。
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N-benzyl-2-chloro-N-[1-(4-morpholin-4-ylbenzoyl)azepan-4-yl]acetamide
CAS number:2143467-62-1 molecular formula:
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| Chinese alias | - | ||
| English alias | - | ||
| CAS number | 2143467-62-1 | molecular formula | |
| molecular weight | 470.000 g/mol | Exact mass | ≥99% |
| PSA | 53.100 Ų | logp | 3.700 |
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