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Tilfrinib

CAS number:1600515-49-8    molecular formula:C17H13N3O

overview

compound introduction

Tilfrinib (化合物 4f) 是一种高效、选择性的 Brk/PTK6 抑制剂,其对 Brk 的 IC50 值为 3.15 nM。Tilfrinib 具有较好的抗增殖活性,有抗肿瘤的潜力。 Product description Tilfrinib (compound 4f) is a potent and selective Brk/PTK6 inhibitor with an IC50 value of 3.15 nM for Brk. Tilfrinib shows good anti-proliferative activity and has potential of anti-tumour.

Specs

Chinese alias3-(9H-吡啶基[2,3-b]吲哚-4-基氨基)苯酚
English alias3-(9H-Pyrido[2,3-b]indol-4-ylamino)phenol
CAS number1600515-49-8molecular formulaC17H13N3O
molecular weight275.3 g/molExact mass≥98%(HPLC)
PSA60.900 Ųlogp3.800

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