CAS number：2556836-50-9 molecular formula：C32H33ClN8O2
Information DGY-06-116 DGY-06-116 is an irreversible covalent and selective inhibitor of Src with IC50 of 2.6 nM. Targets Src (Cell-free assay) 2.6 nM In vitro DGY-06-116 inhibits Src enzymatic activity. DGY-06-116 binds covalently to Src in a manner similar to SM1-71, where the p-loop must kink to establish the covalent bond.
| Chinese alias | - | ||
| English alias | 4-((2-acrylamidophenyl)amino)-N-(2-chloro-6-methylphenyl)-2-((4-(4-methylpiperazin-1-yl)phenyl)amino)pyrimidine-5-carboxamide | ||
| CAS number | 2556836-50-9 | molecular formula | C32H33ClN8O2 |
| molecular weight | 597.11 g/mol | Exact mass | ≥97% |
| PSA | 115.000 Ų | logp | 6.000 |
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