Faldaprevir (BI 201335) 是一种对丙型肝炎病毒 (HCV) 1a 和 1b 基因型的NS3/4A蛋白酶的口服有效的选择性非共价抑制剂,其 Ki值分别为 2.6 和 2.0 nM。Faldaprevir 抑制HCVRNA 复制,其EC50分别为 6.5 和 3.1 nM。Faldaprevir 对慢性HCV感染具有强大的抗病毒活性。
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Faldaprevir
CAS number:801283-95-4 molecular formula:C40H49BrN6O9S
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| Chinese alias | - | ||
| English alias | - | ||
| CAS number | 801283-95-4 | molecular formula | C40H49BrN6O9S |
| molecular weight | 869.8 g/mol | Exact mass | ≥98% |
| PSA | 227.000 Ų | logp | 6.4 |
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