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GW406108X

CAS number:1644443-92-4    molecular formula:C20H11Cl2NO4

overview

compound introduction

应用: GW406108X 是特异性的 Kif15 (Kinesin-12) 抑制剂,IC50 为 0.82 uM。GW406108X 是一种有效的自噬 (autophagy) 抑制剂, ATP 竞争性抑制 ULK1,pIC50 为 6.37 (427 nM)。GW406108X 抑制 ULK1 和自噬,而不影响 mTOR 或 AMPK 活性。

Specs

Chinese alias-
English alias-
CAS number1644443-92-4molecular formulaC20H11Cl2NO4
molecular weight400.21 g/molExact mass≥98%
PSA79.500 Ųlogp4.500

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