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KPLH1130

CAS number:906669-07-6    molecular formula:C15H13N3O3

overview

compound introduction

KPLH1130 是一种丙酮酸脱氢酶激酶 (PDK) 特异性抑制剂,可阻断巨噬细胞极化,减轻炎症反应。KPLH1130 可改善高脂饮食喂养小鼠的葡萄糖耐受性。 KPLH1130 is a specific pyruvate dehydrogenase kinase (PDK) inhibitor, blocks macrophage polarization and attenuates proinflammatory responses. KPLH1130 improves glucose tolerance in HFD-fed mice.

Specs

Chinese alias-
English alias-
CAS number906669-07-6molecular formulaC15H13N3O3
molecular weight283.28 g/molExact mass≥98%
PSA85.200 Ųlogp2.200

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