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ML299

CAS number:1426916-00-8    molecular formula:C23H26BrFN4O2

overview

compound introduction

ML299 是 磷脂酶 D1 和 磷脂酶 D2 的选择性变构调节剂和双重抑制剂 (IC50 值分别为 6 和 12 nM)。ML299 减少 U87-MG 胶质母细胞瘤细胞的侵袭性迁移。 ML299 is a selective allosteric modulator and a dual inhibitor of phospholipases D1 and D2 (IC50 values are 6 and 12 nM, respectively). ML299 decreases invasive migration in U87-MG glioblastoma cells

Specs

Chinese alias-
English aliasVU0463568
CAS number1426916-00-8molecular formulaC23H26BrFN4O2
molecular weight489.38 g/molExact mass≥95%
PSA64.700 Ųlogp3.500

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