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DW14800

CAS number:2243709-60-4    molecular formula:C31H36N4O3

overview

compound introduction

DW14800 is a protein arginine methyltransferase 5 ( PRMT5 ) inhibitor, with an IC 50 of 17 nM. DW14800 reduces H4R3me2s levels and enhances the transcription of HNF4α, but does not alter PRMT5 expression. Anti-cancer activity Form:Solid IC50& Target:PRMT5

Specs

Chinese alias-
English alias-
CAS number2243709-60-4molecular formulaC31H36N4O3
molecular weight512.64 g/molExact mass≥99%
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