compound introduction
[Leu5]-Enkephalin, amide is a δ opioid receptor agonist. In Vitro [Leu5]-Enkephalin causes concentration-dependent, reversible inhibition of pelvic nerve-evoked contractions, with an IC 50 value of 2.1 nM. MCE has not independently confirmed the accuracy of these methods. They are for reference only. In Vivo Levels of [Leu5]-Enkephalin are significantly increased in the nucleus raphe magnus (NRM) of rats 2 weeks after the injection of complete Freund's adjuvant (CFA) (1.02±0.2 pmol/mg protein) as compared with saline-treated rats (0.49±0.04 pmol/mg protein; p Form:Solid IC50& Target:δ opioid receptor
