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2-(1-oxoisoindolin-2-yl)-2-phenyl-N-(thiazol-2-yl)acetamide

CAS number:892772-75-7    molecular formula:C19H15N3O2S

overview

compound introduction

EAI001 是一个有效的选择性突变体表皮生长因子受体 (EGFR) 变构抑制剂,抑制EGFRL858R/T790M的IC50值为 24 nM。EAI001 可用于癌症研究。

Specs

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English alias-
CAS number892772-75-7molecular formulaC19H15N3O2S
molecular weight349.4 g/molExact mass≥99%
PSA90.500 Ųlogp2.900

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