Aditoprime (Aditoprim) 是一种选择性细菌二氢叶酸还原酶(DHFR)抑制剂,可抑制二氢叶酸向四氢叶酸的转化。Aditoprime 抑制大肠杆菌和干酪乳杆菌 DHFR 的 IC50分别为 47 和 520 nM。Aditoprime 具有广谱抗菌、良好的抗菌活性和良好的药代动力学。
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Aditoprime
CAS number:56066-63-8 molecular formula:C15H21N5O2
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| Chinese alias | - | ||
| English alias | - | ||
| CAS number | 56066-63-8 | molecular formula | C15H21N5O2 |
| molecular weight | 303.36 g/mol | Exact mass | ≥99% |
| PSA | 99.500 Ų | logp | 1.500 |
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