ML352 是突触前胆碱转运体(CHT) 的非竞争性抑制剂,对于表达人 CHT 和小鼠前脑突触体的 HEK293细胞,其Ki值分别为 92 nM 和 166 nM。
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N-((3-isopropylisoxazol-5-yl)methyl)-4-methoxy-3-((1-methylpiperidin-4-yl)oxy)benzamide
CAS number:1649450-12-3 molecular formula:C21H29N3O4
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| Chinese alias | - | ||
| English alias | - | ||
| CAS number | 1649450-12-3 | molecular formula | C21H29N3O4 |
| molecular weight | 387.47 g/mol | Exact mass | ≥99% |
| PSA | 76.800 Ų | logp | 2.900 |
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