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5-Tyr-6,8,9-trp-10-arg-neurokinin A (4-10)

CAS number:126050-12-2    molecular formula:C57H68N14O10

overview

compound introduction

MEN 10207 是一种选择性NK-2(Neurokinin Receptor) 速激肽受体拮抗剂。MEN 10207 在 NK-1、NK-2 和 NK-3 速激肽受体的三种单受体体外测定中的 pA2值分别为 5.2、7.9 和 4.9。

Specs

Chinese alias-
English alias-
CAS number126050-12-2molecular formulaC57H68N14O10
molecular weight1109.2 g/molExact mass≥99%
PSA413.000 Ųlogp0.100

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