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BM-1244

CAS number:1619923-32-8    molecular formula:C54H59ClF4N6O8S4

overview

compound introduction

BM-1244 (APG-1252-M1) is a potent Bcl-xL / Bcl-2 inhibitor with K i s of 134 and 450 nM for Bcl- xL and Bcl-2 , respectively. BM-1244 inhibits senescent fibroblasts (SnCs) with an EC 50 of 5 nM. (From patent WO2019033119A1). Form:Solid

Specs

Chinese alias-
English alias-
CAS number1619923-32-8molecular formulaC54H59ClF4N6O8S4
molecular weight1159.79 g/molExact mass≥98%
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