Tubulysin B 是一种高度细胞毒性的肽,有效的微管去稳定剂,是从粘细菌Archangium geophyra和Angiococcus disciformis中分离的。Tubulysin B 抑制许多癌细胞系,包括具有多药抗性的细胞系,IC50值在皮纳摩尔范围内。Tubulysin B 是一种具有细胞毒性活性微管溶素,抑制微管蛋白聚合并导致细胞周期停滞和凋亡。
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Tubulysin B
CAS number:205304-87-6 molecular formula:
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| Chinese alias | - | ||
| English alias | - | ||
| CAS number | 205304-87-6 | molecular formula | |
| molecular weight | 830.000 g/mol | Exact mass | ≥99% |
| PSA | 233.000 Ų | logp | 4.200 |
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