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Tubulysin B

CAS number:205304-87-6    molecular formula:

overview

compound introduction

Tubulysin B 是一种高度细胞毒性的肽,有效的微管去稳定剂,是从粘细菌Archangium geophyra和Angiococcus disciformis中分离的。Tubulysin B 抑制许多癌细胞系,包括具有多药抗性的细胞系,IC50值在皮纳摩尔范围内。Tubulysin B 是一种具有细胞毒性活性微管溶素,抑制微管蛋白聚合并导致细胞周期停滞和凋亡。

Specs

Chinese alias-
English alias-
CAS number205304-87-6molecular formula
molecular weight830.000 g/molExact mass≥99%
PSA233.000 Ųlogp4.200

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