compound introduction
Relacorilant 是一种有效的，选择性的糖皮质激素受体 (glucocorticoid receptor) 拮抗剂，在 HepG2 TAT 实验中，Ki 值为 7.2 nM，在细胞体系中，对大鼠，人和猴子糖皮质激素受体的 Ki 值分别为 12，81.2，210 nM；Relacorilant 有潜力用于库欣综合征的研究。
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Relacorilant
CAS number：1496510-51-0 molecular formula：C27H22N6O3F4S
overview
Specs
| Chinese alias | 雷科瑞兰 | ||
| English alias | Relacorilant | BDBM50265673 | Methanone, ((4aR)-1-(4-fluorophenyl)-1,4,5,6,7,8-hexahydro-6-((1-methyl-1H-pyrazol-4-yl)sulfonyl)-4ah-pyrazolo(3,4-g)isoquinolin-4a-yl)(4-(trifluoromethyl)-2-pyridinyl)- | (R)-(1-(4-fluorophenyl)-6-((1-methyl-1H-pyrazol-4-yl) | ||
| CAS number | 1496510-51-0 | molecular formula | C27H22N6O3F4S |
| molecular weight | 586.6 g/mol | Exact mass | - |
| PSA | 111.000 Ų | logp | 2.9 |
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