compound introduction
RVD-Hpα TFA是一种N-末端延伸的人类加压素，作为选择性CB1受体激动剂。RVD Hpα TFA增加体外表达CB1受体的细胞内Ca2+水平。RVD HpαTFA也是高亲和力CB2阳性变构调节剂（Ki=50nM）。 RVD-Hpα TFA is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. RVD-Hpα TFA increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. RVD-Hpα TFA also high affinity CB2 positive allosteric modulator (Ki=50 nM).
