compound introduction
Yp537 TFA is an estrogen receptor (ER) inhibitor that blocks dimerization of the human estrogen receptor. Appearance:Solid In Vitro:Yp537 TFA (5-50 μM; 1 h) abolishes the formation of the hER-ERE complex. And dose not inhibit the formation of the STAT1-serum-induced element complex. Yp537 TFA binds to a SH2-like domain, and interferes with the SH2-like phosphopeptide coupling mec Biological Activity:Yp537 TFA is an estrogen receptor (ER) inhibitor that blocks dimerization of the human estrogen receptor.
