All
Chemical Reagents
Biomedicine
Organic raw materials
Inorganic chemical industry
intermediate
Agricultural chemicals
Auxiliaries and catalysts
Fragrances and Flavors
Dyes and Pigments
Daily chemical industry

(-)-Indolactam V

CAS number:90365-57-4    molecular formula:C17H23N3O2

overview

compound introduction

(-)-Indolactam V is a PKC activator (Kis: 3.36 nM, 1.03 μM for η-CRD2 , γ-CRD2). (-)-Indolactam V also has the Kds are 5.5 nM (η-C1B), 7.7 nM (ε-C1B), 8.3 nM (δ-C1B), 18.9 nM (β-C1A-long), 20.8 nM (α-C1A-long), 137 nM (β-C1B), 138 nM (γ-C1A), 213 nM (γ-C1B). It has antitumor activity.

Specs

Chinese alias(2S,5S)-1,2,4,5,6,8-六氢-5-(羟甲基)-1-甲基-2-(1-甲基乙基)-3H-吡咯并[4,3,2-gh]-1,4-苯并重氮-3-酮 | (-)-吲哚美坦V | 吲哚内酰胺 V | (2S,5S)-5-(羟甲基)-2-异丙基-1-甲基-4,5,6,8-四氢-1H-[1,4]二氮杂环壬烷并[7,6,5-cd]吲哚-3(2H)-酮
English aliasHY-12307 | MS-24344 | NCGC00345085-01 | (+-)-IL-V | SCHEMBL1278694 | (-)-IndolactamV | CHRYSOPHANIC ACID [WHO-DD] | INDOLACTAM V, (-) | PDSP1_001380 | Indolactam V | AS-17451 | (10S,13S)-13-Hydroxymethyl-10-isopropyl-9-methyl-3,9,12-triaza-tricyclo[6.6.1.
CAS number90365-57-4molecular formulaC17H23N3O2
molecular weight301.38 g/molExact mass-
PSA68.400 Ųlogp2.300

numbering system

No numbering system information yet

physicochemical properties

No physical and chemical property information yet

Safety information

No safety information yet

Production methods and uses

No production method and use information yet

Related

upstream information

No upstream information yet

downstream information

No downstream information yet

MSDS

Found 0 shareMSDS