Ac-IETD-CHO 是一种有效的、可逆的 granzyme B 和 caspase-8 抑制剂。 Ac-IETD-CHO 抑制 Fas 介导的细胞凋亡 (Apoptosis)、出血和肝衰竭。Ac-IETD-CHO还可抑制细胞毒性 T 淋巴细胞诱导的细胞死亡。 Ac-IETD-CHO is a potent, reversible inhibitor of granzyme B and caspase-8. Ac-IETD-CHO inhibits Fas-mediated apoptotic cell death, hemorrhage, and liver failure. Ac-IETD-CHO also inhibits cytotoxic T lymphocytes induced cell death.
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Ac-IETD-CHO
CAS number:191338-86-0 molecular formula:C21H34N4O10
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| Chinese alias | - | ||
| English alias | Granzyme B inhibitor | Ac-IETD-CHO | ||
| CAS number | 191338-86-0 | molecular formula | C21H34N4O10 |
| molecular weight | 502.52 g/mol | Exact mass | ≥95% |
| PSA | 228.000 Ų | logp | -2.000 |
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