CAS number：111011-76-8 molecular formula：C36H45ClN3O8P
外消旋依非替尼具有L型和T型钙通道蛋白抑制剂活性。R（-）异构体似乎对T型钙通道具有很高的选择性。S（+）异构体几乎相等地抑制表达的Ca（V）1.2，Ca（V）1.3和Ca（V）3.1通道电流。 Racemic efonidipine has both L-type and T-type calcium channel protein inhibitor activity. The R(?)-isomer appears to be very selective for T-type calcium channel. The S(+)-isomer inhibits the expressed Ca(V)1.2, Ca(V)1.3 and Ca(V)3.1 channel currents almost equally.
| Chinese alias | - | ||
| English alias | Efonidipine hydrochloride ethanol | NZ 105 ethanolate | EFONIDIPINE HCL MONOETHANOLATE | NZ-105 hydrochloride monoethanolate | CAS-3113-71-1 | AKOS024457778 | SMR003475016 | Landel (TN) | 1,4-trans-cyclohexane diamine | Q27269529 | Efonidipine hydrochlori | ||
| CAS number | 111011-76-8 | molecular formula | C36H45ClN3O8P |
| molecular weight | 714.18 g/mol | Exact mass | 10mM in DMSO |
| PSA | 143.000 Ų | logp | - |
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