CAS number：2222635-15-4 molecular formula：C26H28F3N7O2
DCLK1-IN-1 is a selective, in vivo-compatible chemical probe of the doublecortin like kinase 1 (DCLK1) domain that binds to DCLK1 and DCLK2 with IC50 of 9.5 nM and 31 nM, respectively. DCLK1-IN-1 inhibits DCLK1 and DCLK2 kinases with IC50 of 57.2 nM and 103 nM in kinase assay, respectively.
| Chinese alias | - | ||
| English alias | 5,11-Dihydro-2-[[2-methoxy-4-(4-methyl-1-piperazinyl)phenyl]amino]-11-methyl-5-(2,2,2-trifluoroethyl)-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one | ||
| CAS number | 2222635-15-4 | molecular formula | C26H28F3N7O2 |
| molecular weight | 527.55 g/mol | Exact mass | - |
| PSA | 77.100 Ų | logp | 4.200 |
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