Share to
Overview
Specs
Technical Documents
Related
Articles
reviews
Consult
returns
Product introduction
CEP-28122 mesylate salt 是一种二氨基嘧啶衍生物,是一种高度有效的选择性且具有口服活性的 ALK 抑制剂,对重组 ALK 激酶活性的 IC50 为 1.9 nM。CEP-28122 在人类癌症的 ALK 阳性实验模型中具有抗肿瘤活性。 CEP-28122 具有良好的药效药代活性。 CEP-28122 mesylate salt, a diaminopyrimidine derivative, is a potent, selective, and orally bioavailable ALK inhibitor, with an IC50 value of 1.9 nM for recombinant ALK kinase activity. CEP-28122 has antitumor activity in experimental models of ALK-positive human cancers. CEP-28122 mesylate salt has good pharmacodynamic and pharmacokinetic activity
Chinese name
CEP-28122 mesylate salt , ALK 受体酪氨酸激酶抑制剂
English name
CEP-28122
Chinese alias
-
English alias
(1S,2S,3R,4R)-3-[[5-chloro-2-[[(7S)-4-methoxy-7-morpholin-4-yl-6,7,8,9-tetrahydro-5H-benzo[7]annulen-3-yl]amino]pyrimidin-4-yl]amino]bicyclo[2.2.1]hept-5-ene-2-carboxamide | AC-36009 | CEP 28122 | EX-A1541 | 1431697-87-8 | HY-18030 | Bicyclo[2.2.1]hept-5-
CAS number
2070009-30-0
molecular formula
C29H39ClN6O6S
molecular weight
635.17 g/mol
Exact mass
-
PSA
115.000 Ų
Logp
4.100
Technical Documents
「No technical documents」
Related
「No upstream and downstream information yet」
Articles
「No related articles yet」
user reviews
Loading...
Consultation

Warm reminder:

Because the manufacturer may temporarily adjust product specifications, prices, inventory, parameters and other information without notice, and there are differences in each user's consultation time and procurement needs, the platform reply content is only of reference value within a certain period. Sorry for the inconvenience caused to you, and thank you for your understanding and support! Please consult the online customer service for the latest details. Everything is subject to the real-time reply of the customer service.!

After Sales Services

Please check the quantity, appearance and product information in time when you receive the goods. In case of damage, wrong delivery, abnormal quality and other problems, please feel free to contact us.

Service Hotline:400-6226-992 ,We will handle it for you as soon as possible, thank you for your support and trust.!

Research chemical EP; 25mg; ≥98%

Research chemical EP; 25mg; ≥98%; supplied for laboratory research, analysis, inspection, and scientific procurement use; specifications: EP; 25mg; ≥98%.

item number:C346893-25mg
Product model:25mg
level: EP; 25mg; ≥98%
Lead Time:30days
sold 233 Items
Ask Solution engineer
Specifications:

25mg

Qty

Recommended for you