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Product introduction

DEL-22379 是一种 ERK 二聚化抑制剂。DEL-22379 易与 ERK2 结合，Kd 为低微摩尔水平，即使在低纳摩尔浓度下也可检测到 EL-22379 与 ERK2 结合。DEL-22379 抑制 ERK2 二聚化，IC50 约为 0.5 μM。 application： DEL 22379 is a useful research chemical.DEL 22379 was used for preparation of hydrosoluble 3-arylidene-2-oxyindole tyrosine kinase inhibitors. product description： DEL-22379 is an ERK dimerization Inhibitor. DEL-22379 readily binds to ERK2 with a Kd estimated in the low micromolar range, though binding is detectable even at low nanomolar concentrations. ERK2 dimerization is progressively inhibited with an IC50 of ~0.5 μM.

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Chinese name

DEL 22379

English name

DEL 22379

Chinese alias

N-[2,3-二氢-3-[(5-甲氧基-1H-吲哚-3-基)亚甲基] -2-氧代-1H-吲哚-5-基] -1-哌啶丙烷 | DEL-22379 | N-[2,3-二氢-3-[(5-甲氧基-1H-吲哚-3-基)亚甲基]-2-氧代-1H-吲哚-5-基]-1-哌啶丙酰胺

English alias

CAS number

181223-80-3

molecular formula

C26H28N4O3

molecular weight

444.53 g/mol

Exact mass

10mM in DMSO

PSA

86.500 Å²

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