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Product introduction

EST64454 hydrochloride is a selective and orally active sigma-1 receptor antagonist with a K i of 22 nM. EST64454 hydrochloride has the potential for the research of the pain. In Vivo EST64454 (10 mg/kg; p.o.; male Wistar rats) treatment shows the C max , t 1/2 , AUC 0-∞ , V ss and F% are 771 ng/mL, 3.4 hours, 1431 ng h/mL, 4.4 l/kg and 69%, respectively . EST64454 (10 mg/kg; p.o.; male CD1 mice) treatment shows the C max , t 1/2 , AUC 0-∞ , V ss and F% were 1178 ng/mL, Form:Solid

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Chinese name

EST64454 hydrochloride

English name

EST64454 hydrochloride

Chinese alias

EST64454 盐酸盐

English alias

CAS number

1950569-11-5

molecular formula

C18H23ClF2N4O2

molecular weight

400.85 g/mol

Exact mass

≥99%

PSA

Logp

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